A Phase 1/2 Trial of Multiple Oral Doses of OPC-167832 for Uncomplicated Pulmonary Tuberculosis

PHASE1/PHASE2CompletedINTERVENTIONAL
Enrollment

122

Participants

Timeline

Start Date

October 18, 2018

Primary Completion Date

February 14, 2022

Study Completion Date

March 11, 2022

Conditions
Pulmonary TB
Interventions
DRUG

10 mg OPC-167832

Once daily oral dose of 10 mg OPC-167832 from Day 1 through Day 14.

DRUG

30 mg OPC-167832

Once daily oral dose of 30 mg OPC-167832 from Day 1 through Day 14.

DRUG

90 mg OPC-167832

Once daily oral dose of 90 mg OPC-167832 from Day 1 through Day 14.

DRUG

3 mg OPC-167832

Once daily oral dose of 3 mg OPC-167832 from Day 1 through Day 14.

DRUG

RHEZ

"RHEZ was used in both Stage 1 and Stage 2. Each tablet contains 150 mg rifampicin, 75 mg isoniazid, 400 mg pyrazinamide, and 275 mg ethambutol. Participants received a single-dose from Day 1 through Day 20. The total number of tablets per day was based on the pretreatment body weight:~* Participants weighing 30 to 37 kg received 2 tablets per day~* Participants weighing 38 to 54 kg received 3 tablets per day~* Participants weighing 55 to 70 kg received 4 tablets per day~* Participants weighing \> 70 kg received 5 tablets per day"

DRUG

30 mg OPC-167832 + 300 mg delamanid

Once daily oral dose of 30 mg OPC-167832 plus 300 mg delamanid from Day 1 through Day 14.

DRUG

30 mg OPC-167832 + 400 mg BDQ

Once daily oral dose of 30 mg OPC-167832 plus 400 mg BDQ from Day 1 through Day 14. Participants received a loading dose of 700 mg BDQ on Day 1 and 500 mg on Day 2. The dose of BDQ was 400 mg QD for Days 3 to 14.

DRUG

30 mg OPC-167832 + 300 mg delamanid + 400 mg BDQ

Once daily oral dose of 30 mg OPC-167832 plus 300 mg delamanid plus 400 mg BDQ from Day 1 through Day 14. Participants received a loading dose of 700 mg BDQ on Day 1 and 500 mg on Day 2. The dose of BDQ was 400 mg QD for Days 3 to 14.

Trial Locations (3)

7405

Satellite Site: Task at Brooklyn Chest Hospital, Cape Town

7530

TASK Clinical Research Centre, Cape Town

7700

University of Cape Town (Pty) Ltd., Cape Town

All Listed Sponsors
collaborator

Bill and Melinda Gates Foundation

OTHER

lead

Otsuka Pharmaceutical Development & Commercialization, Inc.

INDUSTRY

NCT03678688 - A Phase 1/2 Trial of Multiple Oral Doses of OPC-167832 for Uncomplicated Pulmonary Tuberculosis | Biotech Hunter | Biotech Hunter