A Study of APG-115 in as a Monotherapy or Combination With Pembrolizumab in Patients With Metastatic Melanomas or Advanced Solid Tumors

PHASE1/PHASE2Active, not recruitingINTERVENTIONAL
Enrollment

230

Participants

Timeline

Start Date

August 29, 2018

Primary Completion Date

December 30, 2025

Study Completion Date

December 30, 2025

Conditions
Unresectable or Metastatic Melanoma or Advanced Solid TumorsMelanomaUveal MelanomaP53 MutationMDM2 Gene MutationCutaneous MelanomaMucosal MelanomaMalignant Peripheral Nerve Sheath Tumors (MPNST)
Interventions
DRUG

Phase 1b: APG-115+pembrolizumab

"dose escalation of APG-115 in combination with label dose of pembrolizumab, Four dose levels of APG-115 will be tested: 50, 100, 150, and 200 mg. APG-115 will be administrateddose escalation of APG-115 in combination with label dose of pembrolizumab, Fourfour dose levels of APG-115 will be tested: 50, 100, 150, and 200 mg. APG-115 will be administrated orally every other day (QOD) for consecutive 2 weeks (ie. dosed at Day 1, 3, 5, 7, 9, 11, and 13), with one week dosing off as there are cycles every 3-weeks a cycle. Pembrolizumab is administrated following FDA approved label dose, i.e., 200 mg intravenous infusion at Day 1 of every 3 weeks as a cycle.~Phase II: Combination of APG-115 at 150 mg (RP2D) and pembrolizumab or APG-115 monotherapy alone."

Trial Locations (21)

4101

Queensland Children's Hospital, South Brisbane

5042

Flinders Medical Centre, Bedford Park

10065

Memorial Sloan Kettering, New York

17033

Penn State Hershey Medical Center Cancer Institute, Hershey

19107

Thomas Jefferson University Hospital, Philadelphia

20010

Children's National Research Institute, Washington D.C.

22031

Virginia Cancer Specialists, Fairfax

27710

Duke Cancer Institute, Durham

33908

Sarah Cannon/FCSRI, Fort Myers

37203

Sarah Cannon Cancer Center, Nashville

44195

Cleveland Clinic, Cleveland

45229

Cincinnati Children's Hospital Medical Center, Cincinnati

63110

Washington University School of Medicine, St Louis

72758

Highlands Oncology, Rogers

77030

University of Texas MD Anderson Cancer Center, Houston

78229

Next Oncology, San Antonio

85724

University of Arizona Cancer Center, Tucson

90095

UCLA Hematology & Oncology Clinic, Los Angeles

90403

Sarcoma Oncology Research Center, Santa Monica

Unknown

Metro South Hospital and Health Services via Princess Alexandra Hospital, Brisbane

Austin Health, Heidelberg

Sponsors
All Listed Sponsors
collaborator

Merck Sharp & Dohme LLC

INDUSTRY

lead

Ascentage Pharma Group Inc.

INDUSTRY

NCT03611868 - A Study of APG-115 in as a Monotherapy or Combination With Pembrolizumab in Patients With Metastatic Melanomas or Advanced Solid Tumors | Biotech Hunter | Biotech Hunter