Dose Finding Study of Nemiralisib (GSK2269557) in Subjects With an Acute Moderate or Severe Exacerbation of Chronic Obstructive Pulmonary Disease (COPD)

PHASE2TerminatedINTERVENTIONAL
Enrollment

943

Participants

Timeline

Start Date

November 28, 2017

Primary Completion Date

January 10, 2019

Study Completion Date

January 10, 2019

Conditions
Pulmonary Disease, Chronic Obstructive
Interventions
DRUG

Placebo ELLIPTA

Placebo will be administered via oral inhalation route once daily in the morning.

DRUG

Nemiralisib ELLIPTA 50 µg

Nemiralisib is a potent and highly selective inhaled PI3Kd inhibitor being developed as an anti-inflammatory for the treatment of inflammatory airways disease. Nemiralisib 50 µg will be administered as a dry powder inhaler via oral inhalation route. In addition, subjects will receive SOC therapy for the index acute moderate or severe exacerbation of COPD.

DRUG

Nemiralisib ELLIPTA 100 µg

Nemiralisib is a potent and highly selective inhaled PI3Kd inhibitor being developed as an anti-inflammatory for the treatment of inflammatory airways disease. Nemiralisib 100 µg will be administered as a dry powder inhaler via oral inhalation route. In addition, subjects will receive SOC therapy for the index acute moderate or severe exacerbation of COPD.

DRUG

Nemiralisib ELLIPTA 250 µg

Nemiralisib is a potent and highly selective inhaled PI3Kd inhibitor being developed as an anti-inflammatory for the treatment of inflammatory airways disease. Nemiralisib 250 µg will be administered as a dry powder inhaler via oral inhalation route. In addition, subjects will receive SOC therapy for the index acute moderate or severe exacerbation of COPD.

DRUG

Nemiralisib ELLIPTA 500 µg

Nemiralisib is a potent and highly selective inhaled PI3Kd inhibitor being developed as an anti-inflammatory for the treatment of inflammatory airways disease. Nemiralisib 500 µg will be administered as a dry powder inhaler via oral inhalation route. In addition, subjects will receive SOC therapy for the index acute moderate or severe exacerbation of COPD.

DRUG

Nemiralisib ELLIPTA 750 µg

Nemiralisib is a potent and highly selective inhaled PI3Kd inhibitor being developed as an anti-inflammatory for the treatment of inflammatory airways disease. Nemiralisib 750 µg will be administered as a dry powder inhaler via oral inhalation route. In addition, subjects will receive SOC therapy for the index acute moderate or severe exacerbation of COPD.

DRUG

Albuterol (Salbutamol) MDI or nebules

Albuterol (Salbutamol) MDI or nebules will be provided to all subjects as a rescue medication.

DRUG

Standard of care therapy

SoC therapy for the index exacerbation is defined as treatment with oral/systemic corticosteroid (prednisone 40 mg/day or equivalent) for 5 days and antibiotic for 7 days. Subjects will receive SoC as prescribed by the Investigator or medically qualified designee. The dose and/or duration of prednisone and/or the antibiotic can be modified according to the Investigator's/medically qualified designee's judgment or according to local country/institution practice.

Trial Locations (161)

1602

GSK Investigational Site, Florida

2000

GSK Investigational Site, Rosario

2145

GSK Investigational Site, Westmead

2250

GSK Investigational Site, Gosford

3016

GSK Investigational Site, Santo Tomé

3168

GSK Investigational Site, Clayton

4000

GSK Investigational Site, San Miguel de Tucumán

4102

GSK Investigational Site, Woolloongabba

5011

GSK Investigational Site, Woodville South

5500

GSK Investigational Site, Mendoza

5600

GSK Investigational Site, San Rafael

6150

GSK Investigational Site, Murdoch

7600

GSK Investigational Site, Mar del Plata

10003

GSK Investigational Site, Cáceres

12203

GSK Investigational Site, Berlin

14467

GSK Investigational Site, Potsdam

16508

GSK Investigational Site, Erie

17007

GSK Investigational Site, Girona

20122

GSK Investigational Site, Milan

21044

GSK Investigational Site, Columbia

21049

GSK Investigational Site, Tradate (VA)

21431

GSK Investigational Site, Incheon

21502

GSK Investigational Site, Geesthacht

23225

GSK Investigational Site, Richmond

23229

GSK Investigational Site, Richmond

23558

GSK Investigational Site, Lübeck

24210

GSK Investigational Site, Abingdon

24411

GSK Investigational Site, Ponferrada (León)

24837

GSK Investigational Site, Schleswig

26006

GSK Investigational Site, Logroño

26505

GSK Investigational Site, Morgantown

27100

GSK Investigational Site, Pavia

28007

GSK Investigational Site, Madrid

28034

GSK Investigational Site, Madrid

28046

GSK Investigational Site, Madrid

28054

GSK Investigational Site, Gastonia

28223

GSK Investigational Site, Pozuelo de Alarcón/Madrid

29303

GSK Investigational Site, Spartanburg

29609

GSK Investigational Site, Brest

30103

GSK Investigational Site, Adairsville

30173

GSK Investigational Site, Hanover

30189

GSK Investigational Site, Woodstock

30202

GSK Investigational Site, Cartagena (Murcia)

32117

GSK Investigational Site, Daytona Beach

33704

GSK Investigational Site, St. Petersburg

34295

GSK Investigational Site, Montpellier

35033

GSK Investigational Site, Rennes

35365

GSK Investigational Site, Daejeon

36608

GSK Investigational Site, Mobile

37024

GSK Investigational Site, Negrar

39770

GSK Investigational Site, Laredo

42100

GSK Investigational Site, Reggio Emilia

44100

GSK Investigational Site, Guadalajara

45070

GSK Investigational Site, Zapopan

45231

GSK Investigational Site, Cincinnati

45459

GSK Investigational Site, Dayton

48013

GSK Investigational Site, Basurto/Bilbao

48231

GSK Investigational Site, Warendorf

48431

GSK Investigational Site, Rheine

54511

GSK Investigational Site, Vandœuvre-lès-Nancy

54907

GSK Investigational Site, Jeonju-si, Jeollabuk-do

56068

GSK Investigational Site, Koblenz

57702

GSK Investigational Site, Rapid City

60389

GSK Investigational Site, Frankfurt am Main

60596

GSK Investigational Site, Frankfurt am Main

63017

GSK Investigational Site, Chesterfield

63301

GSK Investigational Site, Saint Charles

63739

GSK Investigational Site, Aschaffenburg

64020

GSK Investigational Site, Monterrey

64283

GSK Investigational Site, Darmstadt

68134

GSK Investigational Site, Omaha

69004

GSK Investigational Site, Lyon

80907

GSK Investigational Site, Colorado Springs

83022

GSK Investigational Site, Rosenheim

95123

GSK Investigational Site, Catania

96049

GSK Investigational Site, Bamberg

98125

GSK Investigational Site, Messina

153005

GSK Investigational Site, Ivanovo

173008

GSK Investigational Site, Veliky Novgorod

240564

GSK Investigational Site, Râmnicu Vâlcea

300310

GSK Investigational Site, Timișoara

308007

GSK Investigational Site, Belgorod

390039

GSK Investigational Site, Ryazan

394066

GSK Investigational Site, Voronezh

400015

GSK Investigational Site, Cluj-Napoca

410028

GSK Investigational Site, Saratov

410176

GSK Investigational Site, Oradea

432063

GSK Investigational Site, Ulyanovsk

454048

GSK Investigational Site, Chelyabinsk

454106

GSK Investigational Site, Chelyabinsk

603011

GSK Investigational Site, Nizhny Novgorod

614109

GSK Investigational Site, Perm

617507

GSK Investigational Site, Comuna Alexandru Cel Bun

630102

GSK Investigational Site, Novosibirsk

634003

GSK Investigational Site, Tomsk

650000

GSK Investigational Site, Kemerovo

675000

GSK Investigational Site, Blagoveshchensk

700115

GSK Investigational Site, Iași

720284

GSK Investigational Site, Suceava

29406-7108

GSK Investigational Site, Charleston

C1414AIF

GSK Investigational Site, Ciudad Autonoma de Buenos Aires

C1280AEB

GSK Investigational Site, Buenos Aires

C1424BSF

GSK Investigational Site, Buenos Aires

C1425BEN

GSK Investigational Site, Buenos Aires

C1426ABP

GSK Investigational Site, Buenos Aires

M5500CCG

GSK Investigational Site, Mendoza

T6G 2G3

GSK Investigational Site, Edmonton

T8H 0N2

GSK Investigational Site, Sherwood Park

R2H 2A6

GSK Investigational Site, Winnipeg

N8X 5A6

GSK Investigational Site, Windsor

H3T1E2

GSK Investigational Site, Montreal

G1V 4G5

GSK Investigational Site, Québec

J6E 2B4

GSK Investigational Site, Saint-Charles-Borromée

04103

GSK Investigational Site, Leipzig

00133

GSK Investigational Site, Rome

00189

GSK Investigational Site, Rome

1815 JD

GSK Investigational Site, Alkmaar

4818 CK

GSK Investigational Site, Breda

5623 EJ

GSK Investigational Site, Eindhoven

9728 NT

GSK Investigational Site, Groningen

3844 DG

GSK Investigational Site, Harderwijk

1624 NP

GSK Investigational Site, Hoorn

3083 AN

GSK Investigational Site, Rotterdam

3543 AZ

GSK Investigational Site, Utrecht

8025 AB

GSK Investigational Site, Zwolle

15-044

GSK Investigational Site, Bialystok

82-300

GSK Investigational Site, Elblag

31-209

GSK Investigational Site, Krakow

59-300

GSK Investigational Site, Lubin

55-200

GSK Investigational Site, Oława

41-709

GSK Investigational Site, Ruda Śląska

41-200

GSK Investigational Site, Sosnowiec

76-200

GSK Investigational Site, Słupsk

33-100

GSK Investigational Site, Tarnów

030303

GSK Investigational Site, Bucharest

050159

GSK Investigational Site, Bucharest

656 045

GSK Investigational Site, Barnaul

463-707

GSK Investigational Site, Seongnam-si, Gyeonggi-do

02559

GSK Investigational Site, Seoul

136-705

GSK Investigational Site, Seoul

137-701

GSK Investigational Site, Seoul

143-729

GSK Investigational Site, Seoul

150-713

GSK Investigational Site, Seoul

156-755

GSK Investigational Site, Seoul

08003

GSK Investigational Site, Barcelona

03600

GSK Investigational Site, Elda (Alicante)

06800

GSK Investigational Site, Mérida (Badajoz)

03314

GSK Investigational Site, Orihuela (Alicante)

07198

GSK Investigational Site, Palma de Mallorca

07010

GSK Investigational Site, Pama de Mallorca

SE-413 45

GSK Investigational Site, Gothenburg

SE-221 85

GSK Investigational Site, Lund

S40 4AA

GSK Investigational Site, Chesterfield

ML2 0DP

GSK Investigational Site, Wishaw

BB2 3HH

GSK Investigational Site, Blackburn

BD9 6RJ

GSK Investigational Site, Bradford

B15 2GW

GSK Investigational Site, Edgbaston

EH16 4SA

GSK Investigational Site, Edinburgh

L9 7AL

GSK Investigational Site, Liverpool

S5 7AU

GSK Investigational Site, Sheffield

TS19 8PE

GSK Investigational Site, Stockton-on-Tees

Sponsors

Lead Sponsor

All Listed Sponsors
lead

GlaxoSmithKline

INDUSTRY

NCT03345407 - Dose Finding Study of Nemiralisib (GSK2269557) in Subjects With an Acute Moderate or Severe Exacerbation of Chronic Obstructive Pulmonary Disease (COPD) | Biotech Hunter | Biotech Hunter