A Study of GDC-9545 Alone or in Combination With Palbociclib and/or Luteinizing Hormone-Releasing Hormone (LHRH) Agonist in Locally Advanced or Metastatic Estrogen Receptor-Positive Breast Cancer

PHASE1Active, not recruitingINTERVENTIONAL
Enrollment

181

Participants

Timeline

Start Date

November 24, 2017

Primary Completion Date

July 31, 2026

Study Completion Date

July 31, 2026

Conditions
Breast Cancer
Interventions
DRUG

GDC-9545

GDC-9545 will be administered orally, once daily, on Days 1-28 of each 28-day cycle, until disease progression, unacceptable toxicity, withdrawal of consent, or study termination.

DRUG

Palbociclib

Palbociclib will be administered orally, once daily, at the label-recommended dose of 125 mg on Days 1-21 of each 28-day cycle, until disease progression, unacceptable toxicity, withdrawal of consent, or study termination.

DRUG

LHRH Agonist

The LHRH agonist (leuprolide acetate, goserelin acetate, or triptorelin pamoate) will be administered by injection once every 4 weeks on Day 1 of each 28-day cycle, according to the label. The investigator will choose the appropriate LHRH agonist approved for use in breast cancer.

Trial Locations (23)

2010

St Vincent's Hospital Sydney, Darlinghurst

3000

Peter Maccallum Cancer Centre, Melbourne

10065

Memorial Sloan Kettering Cancer Center, New York

28007

Hospital General Universitario Gregorio Maranon, Madrid

28033

Centro Oncologioco MD Anderson Internacional, Madrid

28034

Hospital Universitario Ramón y Cajal, Madrid

28050

Hospital Universitario HM Sanchinarro, Madrid

37204

Vanderbilt University Medical Center, Nashville

46010

Hospital Clinico Universitario de Valencia, Valencia

80045

University of Colorado, Aurora

02115

Massachusetts General Hospital., Boston

02215

Beth Israel Deaconess Medical Center, Boston

Dana Farber Cancer Institute, Boston

410-769

National Cancer Center, Gyeonggi-do

03080

Seoul National University Hospital, Seoul

03722

Severance Hospital, Yonsei University Health System, Seoul

05505

Asan Medical Center, Seoul

06351

Samsung Medical Center, Seoul

08908

ICO L'Hospitalet, L'Hospitalet de Llobregat

08023

Hospital Quiron Barcelona, Barcelona

08035

Hospital Universitari Vall d'Hebron, Barcelona

E1 2ES

Barts Health NHS Trust, London

SM2 5PT

The Royal Marsden Hospital, Suttton

Sponsors

Lead Sponsor

All Listed Sponsors
lead

Genentech, Inc.

INDUSTRY