First-in-Human Study of an Oral Plasmodium Falciparum Plasma Membrane Protein Inhibitor

PHASE1CompletedINTERVENTIONAL
Enrollment

44

Participants

Timeline

Start Date

March 1, 2016

Primary Completion Date

March 9, 2018

Study Completion Date

March 9, 2018

Conditions
Malaria
Interventions
DRUG

SJ733

SJ733 is an oral, novel inhibitor of Plasmodium Falciparum plasma membrane protein PFATP4. It will be administered as a single, multi, or boosted oral dose.

DRUG

Cobicistat

Commercially available cobicistat 150 mg tablets will be used. It will be administered as a single oral dose together with SJ733.

Trial Locations (1)

38105

St. Jude Children's Research Hospital, Memphis

All Listed Sponsors
collaborator

Medicines for Malaria Venture

OTHER

collaborator

Eisai Inc.

INDUSTRY

collaborator

Global Health Innovative Technology Fund

OTHER

lead

St. Jude Children's Research Hospital

OTHER