A Dose Escalation Study Evaluating the Safety and Tolerability of GDC-0032 in Participants With Locally Advanced or Metastatic Solid Tumors or Non-Hodgkin's Lymphoma (NHL) and in Combination With Endocrine Therapy in Locally Advanced or Metastatic Hormone Receptor-Positive Breast Cancer

PHASE1TerminatedINTERVENTIONAL
Enrollment

674

Participants

Timeline

Start Date

March 16, 2011

Primary Completion Date

June 25, 2021

Study Completion Date

June 25, 2021

Conditions
Solid CancersNon-Hodgkin's Lymphoma
Interventions
DRUG

Fulvestrant

Participants will receive fulvestrant 500 milligrams (mg) via intramuscular injection (as per package insert or Summary of Product Characteristics \[SmPC\]) on Days 1 and 15 of Cycle 1, then on Day 1 of each subsequent cycle, until disease progression (Cycle length: 28 days).

DRUG

GDC-0032

Participants will receive GDC-0032 at escalating (Phase I, Stage 1) or fixed (Phase II and Phase I, Stage 2) doses until disease progression. Cycle 1 may be 35 days in length to allow for a 7-day washout following the initial dose; thereafter, GDC-0032 will be administered orally once daily in 28-day cycles.

DRUG

Letrozole

Participants will receive letrozole 2.5 mg orally (as per Package Insert or SmPC) once daily in 28-day cycles until disease progression.

DRUG

Midazolam

Participants will receive midazolam 5 mg (as per Package Insert or SmPC) in hydrochloride syrup on Days 1 and 16 of Cycle 1.

Trial Locations (31)

10065

Memorial Sloan-Kettering Cancer Center, New York

12206

New York Oncology Hematology, P.C., Albany

34232

Sarah Cannon Res Inst; FL, Sarasota

37203

Sarah Cannon Res Inst; TN Onc, Nashville

37204

Vanderbilt Breast Center; Vanderbilt Health Pharmacy, Nashville

37232

Vanderbilt, Nashville

38138

West Cancer Center, Germantown

46010

Hospital Clinico Universitario de Valencia, Valencia

60637

Univ of Chicago, Chicago

63110

Washington University; Division of Oncology, St Louis

73104

Sarah Cannon Res Inst; OK, Oklahoma City

75230

Mary Crowley Cancer Rsch Ctr, Dallas

75246

Baylor Sammons Cancer Center, Dallas

75702

USO - Tyler Cancer Ctr, Tyler

77030

MD Anderson Cancer Center, Houston

85258

TGen Clinical Research Srvs, Scottsdale

85719

University of Arizona Cancer Center, Tucson

92868

University of California Irvine Medical Center, Orange

94109

Sutter Health, San Francisco

94805

Institut Gustave Roussy, Villejuif

95817

UC Davis; Comprehensive Cancer Center, Sacramento

98684

Northwest Cancer Specialists - Vancouver, Vancouver

98902

Yakima Valley Memorial Hospital/North Star Lodge, Yakima

06510

Yale University, New Haven

33901-8101

Florida Cancer Specialists - Fort Myers (New Hampshire Ct), Fort Myers

48201-2013

Barbara Ann Karmanos Cancer Institute, Detroit

02114

Massachusetts General Hospital Cancer Center, Boston

02115

Dana Farber Cancer Inst., Boston

79606-5208

Texas Cancer Center, Abilene

M5G 2M9

University Health Network; Princess Margaret Hospital; Medical Oncology Dept, Toronto

08740

Hospital Univ Vall d'Hebron; Servicio de Oncologia, Sant Andreu de la Barca

Sponsors

Lead Sponsor

All Listed Sponsors
lead

Genentech, Inc.

INDUSTRY